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- Affymax
- Ambit Biosciences
- Ambrx
- Amylin Pharmaceuticals
- Arana Therapeutics
- ARCA biopharma
- ARIUS Research
- ARYx Therapeutics
- Astex Therapeutics
- BioVex
- BioXell
- Bruin Pharmaceuticals
- Cellectis
- CombinatoRx
- Deltanoid Pharmaceuticals
- Diatos
- Evotec
- FivePrime Therapeutics
- Genmab A/S
- Idenix Pharmaceuticals
- Ikaria
- Infinity Pharmaceuticals
- Intercytex
- Ironwood Pharmaceuticals
- KAI Pharmaceuticals
- Kalypsys
- Kereos
- Micromet
- Molecular Insight Pharmaceuticals
- Neuromed Pharmaceuticals
- Novexel
- NPS Pharmaceuticals
- Optimer Pharmaceuticals
- Palatin Technologies
- PharmaMar
- Prana Biotechnology
- Replidyne
- S*BIO
- Sosei
- Speedel Pharmaceuticals
- Synta Pharmaceuticals
- Syntaxin
- Takara Bio
- Theravance
- Tranzyme Pharma
- Trimeris
- Trubion Pharmaceuticals
- ViroPharma
- WILEX
- Xencor
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